醫師介紹

Doctor Introduction

:::

個人介紹

Chiung-Tong Chen
Chiung-Tong Chen

主任

陳炯東 Chiung-Tong Chen

主任
新藥研究與開發、藥物動力學、藥理學、癌症生物學、疾病動物模式
相關連結
學術論文

期刊論文

期刊論文/Journal Paper
(作者群,論文題目,期刊名稱,出版年月,卷號(期別):頁次起迄)
日期
1 (Wei-Sheng Lin)、林慧怡(Lin, Hui-Yi)、(Hao Chan)、(Min-Hsien Wang)、(Ching-Ping Chen)、(Chien-Fu Liao)、(Yu-Jui Kuo)、(Daih-Huang Kuo)、(Jang-Chang Lee)、陳炯東(Chiung-Tong Chen)*、潘敏雄(Min-Hsiung Pan)*,Postfermented Tea Extract Potently Alleviates Glucose Metabolism Disorders In Vitro and In Vivo,ACS Food Science & Technology,2024 Feb,4(2):479-490 2024 . 02
2 (Cheng-Wei Yang)、(Hsing-Yu Hsu)、(Yue-Zhi Lee)、(Jia-Tsrong Jan)、(Sui-Yuan Chang)、(Yi-Ling Lin)、(Ruey-Bing Yang)、(Tai-Ling Chao)、(Jian-Jong Liang)、(Shu-Jing Lin)、(Chun-Che Liao)、(Chih-Shin Chang)、(Huey-Kang Sytwu)、(Ming-Shiu Hung)、陳炯東(Chiung-Tong Chen)、(Shiow-Ju Lee)*,Natural fucoidans inhibit coronaviruses by targeting viral spike protein and host cell furin,BIOCHEMICAL PHARMACOLOGY,2023 Sep,215():1-13 2023 . 09
3 (Mu-Chun Li)、(Mohane Selvaraj Coumar)、(Shu-Yu Lin)、(Yih-Shyan Lin)、(Guan-Lin Huang)、(Chun-Hwa Chen)、(Tzu-Wen Lien)、(Yi-Wen Wu)、(Yen-Ting Chen)、(Ching-Ping Chen)、(Yu-Chen Huang)、(Kai-Chia Yeh)、(Chen-Ming Yang)、(Bikashita Kalita)、(Shiow-Lin Pan)、(Tsu-An Hsu)、(Teng-Kuang Yeh)、陳炯東(Chiung-Tong Chen)、(Hsing-Pang Hsieh)*,Development of Furanopyrimidine-Based Orally Active Third- Generation EGFR Inhibitors for the Treatment of Non-Small Cell Lung Cancer,JOURNAL OF MEDICINAL CHEMISTRY,2023 Feb,66(4):2566-2588 2023 . 02
4 沈冠印(Kuan-Yin Shen)、楊仲翔(Chung-Hsiang Yang)、陳炯東(Chiung-Tong Chen)、何慧敏(Hui-Min Ho)、邱凡峰(Fang-Feng Chiu)、黃瓊儀(Chiung-Yi Huang)、廖浤鈞(Hung-Chun Liao)、徐嘉蔚(Chia-Wei Hsu)、余冠儀(Guann-Yi Yu)、廖經倫(Ching-Len Liao)、陳信偉(Hsin-Wei Chen)、黃明熙(Ming-Hsi Huang)*、劉士任(Shih-Jen Liu)*,Omicron-specific mRNA vaccine induced cross-protective immunity against ancestral SARS-CoV-2 infection with low neutralizing antibodies,JOURNAL OF MEDICAL VIROLOGY,2023 Jan,95(1):1-7 2023 . 01
5 (Ramajayam Kuppusamy)、(Ying-Ting Hsu)、(Yi-Yu Ke)、(Po-Wei Chang)、(Yung-Chiao Chang)、(Hsiao-Fu Chang)、(Pei-Chen Wang)、(Yu-Hao Lin)、(Yu-Chen Huang)、(Teng-Kuang Yeh)、(Jian-Ying Chuang)、(Horace H. Loh)、(Chuan Shih)、陳炯東(Chiung-Tong Chen)、(Shiu-Hwa Yeh)*、(Shau-Hua Ueng)*,Benzo[b]thiophene-2-carboxamides as novel opioid receptor agonists with potent analgesic effect and reduced constipation,EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY,2022 Dec,243():1-18 2022 . 12
6 (Jyh-Der Leu)、(Shih-Ting Lin)、陳炯東(Chiung-Tong Chen)、(C.-Allen Chang)、(Yi-Jang Lee)*,BPR0C261, An Analogous of Microtubule Disrupting Agent D-24851 Enhances the Radiosensitivity of Human Non-Small Cell Lung Cancer Cells via p53-Dependent and p53-Independent Pathways,INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES,2022 Nov,23(22):1-17 2022 . 11
7 (Shu-Yu Lin)、(Ya-Wen Tien)、(Yi-Yu Ke)、(Yung-Chiao Chang)、(Hsiao-Fu Chang)、(Li-Chin Ou)、(Ping-Yee Law)、(Jing-Hua Xi)、(Pao-Luh Tao)、(Horace H. Loh)、(Yu-Sheng Chao)、(Chuan Shih)、陳炯東(Chiung-Tong Chen)、(Shiu-Hwa Yeh)*、(Shau-Hua Ueng)*,Selective and antagonist-dependent µ-opioid receptor activation by the combination of 2-{[2-(6-chloro-3,4-dihydro-1(2H)-quinolinyl)-2-oxoethyl]sulfanyl}-5-phenyl-4,6-(1H,5H)-pyrimidinedione and naloxone/naltrexone,BIOORGANIC CHEMISTRY,2022 Nov,128():1-17 2022 . 11
8 (Yue-Zhi Lee)、(Hsing-Yu Hsu)、(Cheng-Wei Yang)、(Yi-Ling Lin)、(Sui-Yuan Chang)、(Ruey-Bing Yang)、(Jian-Jong Liang)、(Tai-Ling Chao)、(Chun-Che Liao)、(Han-Chieh Kao)、(Jang-Yang Chang)、(Huey-Kang Sytwu)、陳炯東(Chiung-Tong Chen)、(Shiow-Ju Lee)*,The Synergistic Inhibition of Coronavirus Replication and Induced Cytokine Production by Ciclesonide and the Tylophorine-Based Compound Dbq33b,Pharmaceutics,2022 Jul,14(7):1-17 2022 . 07
9 (Chen-Fu Lo)、(Tai-Yu Chiu)、(Yu-Tzu Liu)、(Li-Rung Huang)、(Teng-Kuang Yeh)、(Kuan-Hsun Huang)、(Kuan-Liang Liu)、(Chia-Yu Hsu)、(Ming-Yu Fang)、(Yu-Chen Huang)、(Tsu-An Hsu)、陳炯東(Chiung-Tong Chen)、(Lun Kelvin Tsou)*,Synthesis and Evaluation of Small Molecule Drug Conjugates Harnessing Thioester-Linked Maytansinoids,Pharmaceutics,2022 Jun,14(7):1-19 2022 . 06
10 (Yi-Fan Chen)、(Chien-Huang Wu)、(Li-Hsien Chen)、(Hao-Wei Lee)、(Jinq-Chyi Lee)、(Teng-Kuang Yeh)、(Jang-Yang Chang)*、(Ming-Chen Chou)、(Hui-Ling Wu)、(Yen-Po Lai)、(Jen-Shin Song)、(Kai-Chia Yeh)、陳炯東(Chiung-Tong Chen)、(Chia-Jui Lee)、(Kak-Shan Shia)*、(Meng-Ru Shen)*,Discovery of Potential Neuroprotective Agents against Paclitaxel-Induced Peripheral Neuropathy,JOURNAL OF MEDICINAL CHEMISTRY,2022 Mar,65(6):4767-4782 2022 . 03
11 (Ching-Hua Tsai)、(Tai-Yu Chiu)、陳炯東(Chiung-Tong Chen)、(Chia-Yu Hsu)、(Ya-Ru Tsai)、(Teng-Kuang Yeh)、(Kuan-Hsun Huang)、(Lun Kelvin Tsou)*,Click Chemistry and Multicomponent Reaction for Linker Diversification of Zinc Dipicolylamine-Based Drug Conjugates,Frontiers in Chemistry,2022 Feb,9():1-9 2022 . 02
12 (Jyuhn-Huarng Juang)*、(Chen-Yi Chen)、(Chen-Wei Kao)、(Yu-Wen Huang)、(Tai-Yu Chiu)、陳炯東(Chiung-Tong Chen),Implanted islet mass influences the effects of dipeptidyl peptidase-IV inhibitor LAF237 on transplantation outcomes in diabetic mice,Biomedical Journal,2021 Dec,44(6):s210-s217 2021 . 12
13 (Kai-Chia Yeh)、(Teng-Kuang Yeh)*、(Chung-Yu Huang)、(Chih-Bo Hu)、(Min-Hsien Wang)、(Yu-Wen Huang)、(Ling-Hui Chou)、(Hsuan-Hui Ho)、(Jen-Shin Song)、(Tsu Hsu)、(Weir-Torn Jiaang)、(Yu-Sheng Chao)、陳炯東(Chiung-Tong Chen)*,DBPR108, a novel dipeptidyl peptidase-4 inhibitor with antihyperglycemic activity,LIFE SCIENCES,2021 Aug,278():1-11 2021 . 08
14 (Yang-Bao Miao)、(Kuan-Hung Chen)、陳炯東(Chiung-Tong Chen)、(Fwu-Long Mi)、(Yu-Jung Lin)、(Yen Chang)、(Chi-Shiun Chiang)、(Jui-To Wang)、(Kun-Ju Lin)、(Hsing-Wen Sung)*,A Noninvasive Gut-to-Brain Oral Drug Delivery System for Treating Brain Tumors,ADVANCED MATERIALS,2021 Aug,33(34):1-11 2021 . 08
15 (Yi-Yu Ke)*、(Tzu-Ting Peng)、(Teng-Kuang Yeh)、(Wen-Zheng Huang)、(Shao-En Chang)、(Szu-Huei Wu)、(Hui-Chen Hung)、(Tsu-An Hsu)、(Shiow-Ju Lee)、(Jeng-Shin Song)、(Wen-Hsing Lin)、(Tung-Jung Chiang)、(Jiunn-Horng Lin)、(Huey-Kang Sytwu)、陳炯東(Chiung-Tong Chen)*,Artificial intelligence approach fighting COVID-19 with repurposing drugs,Biomedical Journal,2020 Aug,43(4):355-362 2020 . 08
16 (WAN-NIEN YU)、賴瑩如、馬瑞彣、何其儻、(SHAN-WEI HUNG)、(YU-HSIN CHEN)、陳炯東(Chiung-Tong Chen)、高振益、魏宗德(Tzong-Der Way)*,Citronellol Induces Necroptosis of Human Lung Cancer Cells via TNF-α Pathway and Reactive Oxygen Species Accumulation,IN VIVO,2019 Jul,33(4):1193-1201 2019 . 07
17 (Ying?Ju Lai)、(Wan?Nien Yu)、郭盛助(Sheng-Chu kuo)、(Chi?Tang Ho)、(Chao?Ming Hung)、魏宗德(Tzong-Der Way)*、陳炯東(Chiung-Tong Chen)*,CSC-3436 inhibits TWIST-induced epithelial-mesenchymal transition via the suppression of Twist/Bmi1/Akt pathway in head and neck squamous cell carcinoma,JOURNAL OF CELLULAR PHYSIOLOGY,2019 Jun,234(6):9118-9129 2019 . 06
18 陳煌輝(Huang-Hui Chen)、張欣蕙(Hsin-Huei Chang)、張俊彥(Jang-Yang Chang)、湯雅筑(Ya-Chu Tang)、鄭永齊、林麗梅(Li-Mei Lin)、鄭淑穎(Shu-Ying Cheng)、黃致翔(Chih-Hsiang Huang)、孫嫚梧(Man-Wu Sun)、陳炯東、郭靜娟(Ching-Chuan Kuo)*,Enhanced B-Raf-mediated NRF2 gene transcription and HATs-mediated NRF2 protein acetylation contributes to ABCC1-mediated chemoresistance and glutathione-mediated survival in acquired topoisomerase II poison-resistant cancer cells,FREE RADICAL BIOLOGY AND MEDICINE,2017 Dec,113():505-518 2017 . 12

研討會論文

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專書

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研究計畫

研究計畫/Research Grant
(研究類型,研究計畫代號,主持人,補助或委託單位名稱,計畫名稱,計畫期間)
日期
1 個別型,NSTC 113-2639-E-007-001-ASP,糜福龍、林昆儒、陳炯東(Chiung-Tong Chen),國科會,非侵入性經腸道直達腦部口服遞送系統(4/5),2024.8.1~2025.7.31 2024 . 08
2 個別型,MOST 111-2320-B-400-007-MY3,陳炯東(Chiung-Tong Chen),國科會,開發臨床PI3K/mTOR標靶藥物合併一可降解Myc致癌蛋白質的新穎激酶抑制劑在癌症的精準治療策略,2024.8.1~2025.7.31 2024 . 08

專利技術

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獲獎事蹟

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技術轉移

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